Bibliografía básica Camille Georges Wermuth (2008). The practice of medicinal chemistry, 3rd Ed. Amsterdam: Elsevier
Camille Georges Wermuth (2014). The practice of medicinal chemistry, 4th Ed. Amsterdam: Elsevier
Graham L. Patrick (2013). An introduction to medicinal chemistry, 5th Ed. Oxford: Oxford University Press

O libro "The practice of medicinal chemistry" 4th Ed. de Camille G. Wermuth está dispoñible on line na web da biblioteca da facultade.

Bibliografía complementaria E. J. Corey, B. Czakó, L. Kürti (2007). Molecules and medicine. New Jersey: John Wiley and Sons
K. C. Nicolaou, T. Montagnon, Eds. (2008). Molecules that changed the world. Weinheim: Wiley-VCH
Edward R. Zartler & Michael J. Shapiro, Eds. (2008). Fragment-based drug discovery, a practical approach. Chichester: John Wiley & Sons
Celerino Abad Zapatero (2013). Ligand efficiency indices for drug discovery. Amsterdam: Elsevier